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Pubblicazioni scientifiche

Anno: 2017

  1. Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
    Pubblicato su: Journal of Enzyme Inhibition and Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Synthesis; biological evaluation and quantitative structure-active relationships of 1;3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2016

  1. Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1;3-thiazolidin-4-one derivatives
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Novel 1;3-thiazolidin-4-one derivatives as promising anti- Candida agents endowed with anti-oxidant and chelating properties
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2015

  1. Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori; anti-malarial and anti-leishmanial agents
    Pubblicato su: Journal of Enzyme Inhibition and Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2014

  1. Design; synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors
    Pubblicato su: Bioorganic and Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2013

  1. Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2012

  1. CPTH6; a thiazole derivative; induces histone hypoacetylation and apoptosis in human leukemia cells
    Pubblicato su: Clinical Cancer Research
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
    Pubblicato su: Current Topics in Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  3. Synthesis; anti-Candida activity; and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2011

  1. Synthesis and biological evaluation of novel 2;4-disubstituted-1;3- thiazoles as anti-Candida spp. agents
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2010

  1. Synthesis and characterization of new 3-acyl-7-hydroxy-6;8-substituted- coumarin and 3-acyl-7-benzyloxy-6;8-substituted-coumarin derivatives
    Pubblicato su: Journal of Heterocyclic Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl) thiazol-2-ylhydrazone derivatives
    Pubblicato su: Journal of Heterocyclic Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  3. Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3;5-di(hetero)aryl-4;5-dihydro-(1H)-pyrazole derivatives
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  4. Synthesis; selective anti-Helicobacter pylori activity; and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2009

  1. Synthesis and biological evaluation of novel conjugated coumarin-thiazole systems
    Pubblicato su: Journal of Heterocyclic Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone.
    Pubblicato su: Journal of medicinal chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  3. Synthesis; molecular modeling; and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins
    Pubblicato su: Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  4. Synthesis and evaluation of 4-acyl-2-thiazolylhydrazone derivatives for anti-Toxoplasma efficacy in vitro
    Pubblicato su: Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2007

  1. A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2006

  1. Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2005

  1. Synthesis and in vitro selective anti-Helicobacter pylori activity of pyrazoline derivatives
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2002

  1. Inhibition of amine oxidases activity by 1-acetyl-3;5-diphenyl-4;5-dihydro-(1H)-pyrazole derivatives
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 2001

  1. Efficacy of Hypericum and Calendula oils in the epithelial reconstruction of surgical wounds in childbirth with caesarean section
    Pubblicato su: Farmaco
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'
  2. Selective inhibition of FAD and copper-dependent amine oxidases by N-acetyl pyrazole derivatives
    Pubblicato su: Inflammation Research
    - Vedi su: 'Scopus'

Anno: 2000

  1. Synthesis and preliminary biological evaluation of 4;6-disubstituted 3-cyanopyridin-2(1H)-ones; a new class of calcium entry blockers
    Pubblicato su: Bioorganic and Medicinal Chemistry Letters
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 1999

  1. Anti-inflammatory; analgesic and antipyretic 4;6-disubstituted 3-cyano- 2-aminopyridines
    Pubblicato su: European Journal of Medicinal Chemistry
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 1998

  1. Inhibitory effect of 1;3;5-triphenyl-4;5-dihydro-(1H)-pyrazole derivatives on activity of amine oxidases
    Pubblicato su: Journal of Enzyme Inhibition
    - Vedi su: 'Scopus'
    - Vedi su: 'ScienceDirect'

Anno: 1996

  1. Synthesis and β-adrenoreceptor blocking activity of [[3-(alkylamine)-2-hydroxypropyl]oximino]pyridines and O[3-(alkylamine)-2-hydroxypropyl]methylpyridine ketone oximes derivatives
    Pubblicato su: Farmaco
    - Vedi su: 'Scopus'

Anno: 1992

  1. Beta-Blocking Pyridin-oximino derivatives
    Pubblicato su: Pharmacological Research
    - Vedi su: 'Scopus'

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