Accesso negato
Pubblicazioni scientifiche
Anno: 2017
-
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
Pubblicato su: Journal of Enzyme Inhibition and Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis; biological evaluation and quantitative structure-active relationships of 1;3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2016
-
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1;3-thiazolidin-4-one derivatives
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Novel 1;3-thiazolidin-4-one derivatives as promising anti- Candida agents endowed with anti-oxidant and chelating properties
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2015
-
Bioactive compounds of Crocus sativus L. and their semi-synthetic derivatives as promising anti-Helicobacter pylori; anti-malarial and anti-leishmanial agents
Pubblicato su: Journal of Enzyme Inhibition and Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2014
-
Design; synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors
Pubblicato su: Bioorganic and Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2013
-
Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2012
-
CPTH6; a thiazole derivative; induces histone hypoacetylation and apoptosis in human leukemia cells
Pubblicato su: Clinical Cancer Research- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
Pubblicato su: Current Topics in Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis; anti-Candida activity; and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2011
-
Synthesis and biological evaluation of novel 2;4-disubstituted-1;3- thiazoles as anti-Candida spp. agents
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2010
-
Synthesis and characterization of new 3-acyl-7-hydroxy-6;8-substituted- coumarin and 3-acyl-7-benzyloxy-6;8-substituted-coumarin derivatives
Pubblicato su: Journal of Heterocyclic Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl) thiazol-2-ylhydrazone derivatives
Pubblicato su: Journal of Heterocyclic Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3;5-di(hetero)aryl-4;5-dihydro-(1H)-pyrazole derivatives
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis; selective anti-Helicobacter pylori activity; and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2009
-
Synthesis and biological evaluation of novel conjugated coumarin-thiazole systems
Pubblicato su: Journal of Heterocyclic Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
A novel histone acetyltransferase inhibitor modulating Gcn5 network: cyclopentylidene-[4-(4'-chlorophenyl)thiazol-2-yl)hydrazone.
Pubblicato su: Journal of medicinal chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis; molecular modeling; and selective inhibitory activity against human monoamine oxidases of 3-carboxamido-7-substituted coumarins
Pubblicato su: Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis and evaluation of 4-acyl-2-thiazolylhydrazone derivatives for anti-Toxoplasma efficacy in vitro
Pubblicato su: Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2007
-
A novel class of selective anti-Helicobacter pylori agents 2-oxo-2H-chromene-3-carboxamide derivatives
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2006
-
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2005
-
Synthesis and in vitro selective anti-Helicobacter pylori activity of pyrazoline derivatives
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2002
-
Inhibition of amine oxidases activity by 1-acetyl-3;5-diphenyl-4;5-dihydro-(1H)-pyrazole derivatives
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 2001
-
Efficacy of Hypericum and Calendula oils in the epithelial reconstruction of surgical wounds in childbirth with caesarean section
Pubblicato su: Farmaco- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect' -
Selective inhibition of FAD and copper-dependent amine oxidases by N-acetyl pyrazole derivatives
Pubblicato su: Inflammation Research- Vedi su: 'Scopus'
Anno: 2000
-
Synthesis and preliminary biological evaluation of 4;6-disubstituted 3-cyanopyridin-2(1H)-ones; a new class of calcium entry blockers
Pubblicato su: Bioorganic and Medicinal Chemistry Letters- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 1999
-
Anti-inflammatory; analgesic and antipyretic 4;6-disubstituted 3-cyano- 2-aminopyridines
Pubblicato su: European Journal of Medicinal Chemistry- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 1998
-
Inhibitory effect of 1;3;5-triphenyl-4;5-dihydro-(1H)-pyrazole derivatives on activity of amine oxidases
Pubblicato su: Journal of Enzyme Inhibition- Vedi su: 'Scopus'
- Vedi su: 'ScienceDirect'
Anno: 1996
-
Synthesis and β-adrenoreceptor blocking activity of [[3-(alkylamine)-2-hydroxypropyl]oximino]pyridines and O[3-(alkylamine)-2-hydroxypropyl]methylpyridine ketone oximes derivatives
Pubblicato su: Farmaco- Vedi su: 'Scopus'
Anno: 1992
-
Beta-Blocking Pyridin-oximino derivatives
Pubblicato su: Pharmacological Research- Vedi su: 'Scopus'